Actim (10mg) 14 Tablets

Bisoprolol 10mg Tablet primarily works by selectively blocking beta-1 adrenergic receptors in the heart and other tissues. This mechanism of action is crucial in its ability to reduce heart rate and lower blood pressure. By blocking these receptors, bisoprolol inhibits the effects of catecholamines, such as adrenaline, on the heart. This leads to a decrease in cardiac output, heart rate, and contractility, resulting in reduced myocardial oxygen demand. Consequently, it helps in the management of hypertension and certain cardiovascular conditions by controlling the heart's response to stress and exertion.

bisoprolol 10mg

Beta-blocker

Tablet

The following are the uses of bisoprolol 10mg Tablet:

• Used for treating high blood pressure, helping to lower and control it.
• Used to manage chest pain (angina) by reducing the frequency and severity of attacks.
• Used to improve survival rates and reduce hospital admissions for heart failure.
• Used to relieve symptoms associated with heart rhythm disorders.
• Used to prevent migraines by reducing their frequency and intensity.
• Used to enhance the effectiveness of other heart medications.
• Used as a long-term treatment option for maintaining heart health.

Tailoring Treatment for Optimal Health, Prescribed Medication Dosage is:

• For high blood pressure (Hypertension)- Start with 2.5-5 mg once daily.
• For chronic heart failure (CHF)- Start with 1.25-5 mg once daily. May increase up to 10 mg once daily if necessary.
• For angina (chest pain due to lack of blood to the heart)- Start with 2.5-5 mg once daily. May increase your dose, depending on your tolerance and response.
• For migraine- The starting dose is 2.5 mg once daily. You may increase your dose, depending on your tolerance and response.

In the case of an overdose of Bisoprolol 10mg tablets, individuals may experience symptoms such as severe dizziness, extreme fatigue, and a significant drop in blood pressure, leading to potential fainting or even cardiac arrest. This medication, when taken in excess, can result in a dangerously slow heart rate and impaired heart function. It is crucial to seek immediate medical assistance if an overdose is suspected, as prompt treatment can prevent severe complications and ensure the well-being of the individual.

In the case of a missed dose of bisoprolol 10mg Tablet, it is important to take the medication as soon as you remember. However, if it is almost time for your next scheduled dose, skip the missed dose and continue with your regular dosing schedule. Do not take a double dose to make up for the missed one. If you miss multiple doses, contact your healthcare provider for guidance on how to adjust your dosing schedule and ensure the effectiveness of the medication. It is crucial to maintain a consistent routine when taking bisoprolol to maximize its benefits.

To take Bisoprolol 10mg Tablet, swallow the tablet whole with a glass of water, preferably in the morning, as directed by your healthcare provider, without crushing or chewing it.

Here are the conditions or situations when Bisoprolol 10mg Tablet should not be used:

• Should not be used in patients with a known allergy or hypersensitivity to Bisoprolol or other beta-blockers.
• Contraindicated in patients with severe bradycardia (very slow heart rate).
• Not suitable for individuals with cardiogenic shock or decompensated heart failure.
• Should not be used in patients with severe hypotension (very low blood pressure).
• Contraindicated during episodes of bronchial asthma or severe bronchospasm.
• Not recommended for patients with severe peripheral arterial disease.
• Should be avoided in individuals with severe renal impairment or kidney failure.
• Not suitable for patients with metabolic acidosis.
• Should not be used during pregnancy or breastfeeding without medical advice.

The side effects of Bisoprolol 10mg Tablet may include:

• Fatigue and weakness
• Dizziness or lightheadedness
• Headache
• Nausea and vomiting
• Diarrhea or constipation
• Cold extremities (hands and feet)
• Slow heart rate (bradycardia)
• Impaired sexual function

Following are the precautions and warnings for Bisoprolol 10mg Tablet:

• This medication is not recommended for individuals with known hypersensitivity or allergy to bisoprolol or any other beta-blockers.
• Patients with a history of respiratory issues like asthma, chronic obstructive pulmonary disease (COPD), or severe bronchitis should exercise caution, as bisoprolol may exacerbate these conditions.
• Bisoprolol can cause low blood pressure and slow heart rate, hence close monitoring is required in patients with existing cardiovascular issues.
• It may mask the symptoms of hypoglycemia, especially in diabetic patients. Regular blood glucose monitoring is advised.
• Caution is advised in patients with peripheral vascular disease, as bisoprolol may aggravate symptoms of poor circulation.
• Patients with a history of kidney or liver problems should be monitored regularly, as bisoprolol is primarily metabolized in these organs.
• Bisoprolol may cause dizziness or fatigue; patients should be cautious when driving or operating heavy machinery.

Following are the drug interactions for Bisoprolol 10mg Tablet:

• Drugs that block the action of adrenaline (beta-blockers) may have an additive effect with bisoprolol, leading to excessive slowing of heart rate and a decrease in blood pressure.
• Bisoprolol can interact with calcium channel blockers, such as verapamil and diltiazem, which may cause a significant drop in heart rate and blood pressure.
• The effect of bisoprolol may be reduced by non-steroidal anti-inflammatory drugs (NSAIDs) like ibuprofen, potentially requiring higher bisoprolol doses.
• Antihypertensive effects of bisoprolol can be reduced by corticosteroids, necessitating close monitoring.
• Antihistamines, when used with bisoprolol, may result in increased heart rate and blood pressure.
• Rifampicin, a strong enzyme inducer, can decrease the effectiveness of bisoprolol by enhancing its metabolism.
• The combination of bisoprolol and digoxin may increase the risk of bradycardia (slow heart rate) and heart block. Close monitoring is advised.
• Concomitant use of bisoprolol and insulin or oral hypoglycemic agents may mask the symptoms of hypoglycemia, such as tremor and increased heart rate.

Following are the food interactions for Bisoprolol 10mg Tablet:

• Grapefruit and grapefruit juice consumption should be avoided as they can increase the levels of bisoprolol in the blood, leading to potential side effects.
• Alcohol intake should be limited as it may reduce the effectiveness of bisoprolol and can cause excessive dizziness and lightheadedness.
• Caffeine-rich beverages like coffee and energy drinks might interact with bisoprolol, affecting heart rate and blood pressure.
• Salt and salty foods should be reduced as bisoprolol is used to manage blood pressure, and high salt intake can counteract its effects.
• Avoid or limit high-potassium foods like bananas, oranges, and tomatoes if you have kidney problems, as bisoprolol can raise potassium levels.
• Licorice can decrease the effectiveness of bisoprolol, so it's best to avoid it while on this medication.
• Always follow your healthcare provider's dietary recommendations to ensure the medication's optimal performance.
• Inform your doctor about any dietary supplements or herbal remedies you're taking to prevent potential interactions.

Bisoprolol 10mg Tablets should be stored in a secure and dry location, preferably at room temperature, away from direct sunlight, heat, and moisture. It is crucial to keep the tablets in their original container, tightly sealed, to maintain their integrity and prevent exposure to environmental factors. Ensure you regularly check the expiration date, and if the medication has passed its expiry, do not use it and dispose of it appropriately. Proper disposal methods are essential; do not flush the tablets or throw them into the trash. Contact your pharmacist or a healthcare professional for guidance on how to safely dispose of unused or expired bisoprolol tablets. Keep this medication out of children's reach to prevent accidental consumption.

Following are the quick tips for Bisoprolol 10mg Tablet:

• Take the tablet as directed by your doctor, typically once daily at the same time each day.
• Swallow the tablet whole with a glass of water, do not crush or chew.
• Do not skip doses, even if you feel well, to maintain consistent blood levels.
• If you forget a dose, take it as soon as you remember, unless it's almost time for your next dose.
• Avoid sudden discontinuation; consult your doctor for instructions on stopping the medication.
• Store the tablets at room temperature, away from moisture and heat.
• Inform your doctor about all medications you're taking to avoid potential interactions.

Lab tests are not required when taking Bisoprolol, however, it is important to regularly monitor your blood pressure and heart rate to ensure the medication is working effectively and to minimize any unwanted side effects. It is recommended that you discuss with a healthcare professional, such as your doctor or pharmacist, the frequency and extent of monitoring to ensure it is personalized to your condition and individual needs. Disclosure of all current medications is important, including herbal supplements and over-the-counter drugs, to ensure no negative interactions occur and to ensure the safety of your medication regime. It is also crucial to keep appointments with your healthcare providers to assess your progress and overall health while on Bisoprolol. During these appointments, any concerns can be addressed through communication with your healthcare team.