SMUR (50mg) 30 Tablets

Eperisone HCl 50mg Tablet primarily acts as a central nervous system (CNS) depressant and a muscle relaxant. Its mechanism of action involves multiple pathways. Firstly, it targets the spinal cord and suppresses polysynaptic reflexes, thereby reducing muscle spasticity. Eperisone inhibits the release of excitatory neurotransmitters, such as glutamate and aspartate, which play a crucial role in muscle contraction and spasticity. By modulating these neurotransmitters, the drug helps in relaxing skeletal muscles. Additionally, Eperisone may enhance the activity of inhibitory neurotransmitters like gamma-aminobutyric acid (GABA), further contributing to its muscle relaxant effect. This multifaceted mechanism makes Eperisone HCl effective in managing various conditions associated with muscle stiffness and pain.

Eperisone HCl 50mg

Muscle relaxant.

Tablet

The following are the uses of Eperisone HCl 50mg Tablet:

• Used for relieving muscle pain and stiffness, especially in conditions like back pain, neck pain, and muscle spasms.
• Used for improving muscle movement and flexibility, aiding in physical therapy and rehabilitation.
• Used for treating muscle spasms associated with certain neurological disorders.
• Used for managing muscle discomfort and tightness in sports injuries and exercise-related soreness.
• Used for providing relief from muscle-related headaches and jaw pain.
• Used for easing muscle-induced discomfort in various musculoskeletal disorders.
• Used for supporting overall muscle relaxation and comfort.

Tailoring Treatment for Optimal Health, Prescribed Medication Dosage is:

• Eperisone Hydrochloride 50mg is usually taken in doses of two tablets per day.
• The dosage may be higher for those with severe disease and should not exceed 6 tablets per day in divided doses.
• It is important to only take the drug when experiencing an active spasm and to stop taking it when symptoms improve to avoid dependence.

In the case of an overdose of Eperisone HCl 50mg Tablets, the severity of symptoms can vary. Individuals may experience heightened muscle relaxation, leading to excessive weakness and difficulty in maintaining posture. Gastrointestinal discomfort, including nausea and stomach pain, might occur. In more serious cases, respiratory depression, a potentially life-threatening condition, can develop. Prompt medical intervention is necessary to manage these symptoms and prevent further complications.

In the case of a missed dose of Eperisone HCl 50mg Tablet, it is important to take the medication as soon as you remember. However, if it is almost time for your next scheduled dose, skip the missed dose and continue with your regular dosing schedule. Do not double the dose to make up for a missed one, as this may increase the risk of side effects. It is recommended to set a daily reminder or keep the medication in a visible place to help you remember to take it as prescribed. Consult your healthcare provider if you frequently miss doses or have concerns about managing your medication schedule.

To take Eperisone HCl 50mg Tablet, swallow the tablet whole with a glass of water, preferably with or after a meal, exactly as prescribed by your healthcare professional, typically 3 times a day or as directed.

Eperisone HCl 50mg tablet should not be used in the following conditions:

• Hypersensitivity or allergy to eperisone hydrochloride or any other ingredients in the tablet.
• Pregnancy or breastfeeding unless prescribed by a healthcare provider, as the safety of eperisone in these conditions has not been fully established.
• Severe liver impairment or liver disease, as eperisone is metabolized in the liver.
• Myasthenia gravis or other conditions that cause muscle weakness, as eperisone is a muscle relaxant and may worsen symptoms.
• In combination with medications that depress the central nervous system, unless recommended by a healthcare provider.

The side effects of Eperisone HCl 50mg Tablet may include:

• Drowsiness or sleepiness
• Nausea and vomiting
• Dry mouth
• Constipation
• Blurred vision
• Dizziness
• Allergic reactions (skin rash, itching)
• Muscle weakness

Following are the precautions and warnings for Eperisone HCl 50mg Tablet:

• Do not take this medication if you are allergic to Eperisone or any other muscle relaxant.
• Patients with liver or kidney disease should exercise caution and consult a doctor, as dosage adjustments may be necessary.
• Avoid driving or operating heavy machinery as this medication may cause dizziness or sleepiness.
• Elderly patients may be more sensitive to the side effects, hence medical supervision is advised.
• Avoid alcohol consumption while taking this medication as it may intensify adverse effects.
• Inform your doctor about all medications you are currently taking to avoid potential drug interactions.
• This medication should be used with caution during pregnancy and breastfeeding, only if the potential benefits outweigh the risks.

Following are the drug interactions for Eperisone HCl 50mg Tablet:

• Eperisone may interact with other central nervous system (CNS) depressants like opioids, benzodiazepines, or alcohol, enhancing their effects and potentially causing excessive sedation or respiratory depression.
• Anticoagulants such as warfarin or heparin may have their effects potentiated, increasing the risk of bleeding.
• The efficacy of neuromuscular blocking agents can be affected by Eperisone, leading to prolonged muscle relaxation during surgery.
• Caution is advised when combining with other muscle relaxants, as it may result in additive effects and increased muscle weakness.
• Drugs that inhibit CYP2C19, such as omeprazole or fluoxetine, may increase Eperisone levels in the body, potentially leading to enhanced side effects.
• Eperisone can decrease the absorption of levodopa, reducing its effectiveness in treating Parkinson's disease.
• Concomitant use with anticholinergic medications may increase the risk of urinary retention and other anticholinergic side effects.

Following are the food interactions to consider with Eperisone HCl 50mg Tablet:

• Avoid grapefruit and grapefruit juice as they may interfere with the metabolism of the medication, potentially increasing its levels in the body and leading to a higher risk of side effects.
• Limit alcohol consumption as it may enhance the sedative effects of Eperisone, causing increased drowsiness and dizziness.
• Fatty meals can slow down the absorption of Eperisone, potentially reducing its effectiveness, so it's best to take the medication on an empty stomach or with a light meal.
• Caffeine intake should be monitored as it may counteract the muscle relaxant effect of Eperisone, reducing its therapeutic benefit.
• Avoid herbal supplements like St. John's Wort, as they can affect the way the body metabolizes Eperisone, potentially reducing its efficacy.
• Consuming high-fiber foods can potentially decrease the absorption of Eperisone, so it is advisable to maintain a consistent diet during the medication course.
• Always follow the dosing instructions provided by your healthcare professional, and inform them about any dietary habits or supplements you are taking.

Eperisone HCl 50mg Tablets should be stored in a secure and dry location, away from direct sunlight and moisture. Maintain the tablets in their original packaging, tightly sealed, to ensure their integrity and prevent contamination. It is crucial to keep the medication away from heat sources like heaters or ovens, as temperature fluctuations can impact its effectiveness. Regularly check the expiration date, and if the tablets are past their prime, proper disposal is essential. Avoid flushing or pouring them down the drain; instead, consult a pharmacist or healthcare professional for safe disposal instructions. Always store medications in a safe place, out of the reach of children, to prevent accidental consumption.

Following are the quick tips for Eperisone HCl 50mg Tablet:

• Take the tablet as directed by your doctor; do not crush or chew it.
• Ensure you complete the full course of medication as prescribed.
• Maintain a consistent time for taking the tablet daily.
• If you experience stomach discomfort, consider taking the tablet with food.
• Avoid consuming alcohol while on this medication.
• Inform your doctor about any other medications you are taking.
• Store the tablets in a cool, dry place, away from direct sunlight.
• Do not share this medication with others, even if their symptoms are similar.

Eperisone Hydrochloride is a muscle relaxant prescribed to patients with spinal cord damage who experience muscle spasms and associated pain. While the medication relieves muscle spasms, it's a strong drug that requires routine laboratory testing to monitor for toxicity and adverse effects on various physiological parameters. This lab work ensures the medication is dosed properly and identifies potential harmful side effects. The lab tests required depend on the patient and doctor preferences. Nevertheless, tests like full blood counts, kidney function tests, and liver function tests are common. It's critical to note that these are examples, and your doctor will determine the appropriate tests. Attending all appointments with your doctor ensures your treatment plan stays on track and addresses any side effects.